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Nuclear Medicine and Biology
Volume 37, Issue 2
, Pages 167-178
, February 2010
Preparation and in vivo evaluation of radioiodinated closo-decaborate(2-) derivatives to identify structural components that provide low retention in tissues
References
- . Alpha-particle radioimmunotherapy with astatine-211 and bismuth-213. Eur J Nucl Med Mol Imaging. 2008;35:1729–1733
- . Targeted alpha-particle radiotherapy with 211At-labeled monoclonal antibodies. Nucl Med Biol. 2007;34:779–785
- . The promise of targeted alpha-particle therapy. J Nucl Med. 2005;46(Suppl 1):199S–204S
- Cancer radioimmunotherapy with alpha-emitting nuclides. Eur J Nucl Med Mol Imaging. 2005;32:601–614
- . Advancements in cancer therapy with alpha-emitters: a review. Int J Rad Oncol Biol Phys. 2001;51:271–278
- . Targeted alpha-therapy: past, present, future?. Dalton Trans. 2007;4918–4928
- . Radiohalogenation of proteins: an overview of radionuclides, labeling methods, and reagents for conjugate labeling. Bioconjug Chem. 1992;3:433–470
- . The synthesis of radiolabeled compounds via organometallic intermediates. Tetrahedron. 1989;45:6601–6621
- . Regiospecific incorporation of no-carrier-added radiobromine and radioiodine into aromatic rings via halogenodegermylation. J Chem Soc Perkin Trans I. 1985;1687–1692
- . [211At]Astatine-labeled compound stability: issues with released [211At]astatide and development of labeling reagents to increase stability. Curr Radiopharm. 2008;1:144–176
- . Reagents for astatination of biomolecules: 2. Conjugation of anionic boron cage pendant groups to a protein provides a method for direct labeling that is stable to in vivo deastatination. Bioconjug Chem. 2007;18:1226–1240
- Reagents for astatination of biomolecules: comparison of the in vivo distribution and stability of some radioiodinated/astatinated benzamidyl and nido-carboranyl compounds. Bioconjug Chem. 2004;15:203–223
- . Biotin reagents in antibody pretargeting: 6. Synthesis and in vivo evaluation of astatinated and radioiodinated aryl- and nido-carboranyl-biotin derivatives. Bioconjug Chem. 2004;15:601–616
- . Synthesis, radioiodination, and biodistribution of some nido- and closo-monocarbon carborane derivatives. Nucl Med Biol. 2004;31:523–530
- Comparative metabolism and retention of iodine-125, yttrium-90, indium-111 radioimmunoconjugates by cancer cells. Cancer Res. 1996;56:2123–2129
- . Intracellular metabolism of indium-111-DTPA-labeled receptor targeted proteins. J Nucl Med. 1993;34:1728–1738
- . Effects of radiolabeling monoclonal antibodies with a residualizing iodine radiolabel on the accretion of radioisotope in tumors. Cancer Res. 1995;55:3132–3139
- . Applications of radiolabeled boron clusters to the diagnosis and treatment of cancer. Chem Rev. 1999;99:3421–3434
- The chemistry of neutron capture therapy. Chem Rev. 1998;98:1515–1562
- . Renal uptake and metabolism of radiopharmaceuticals derived from peptides and proteins. Adv Drug Deliv Rev. 2008;60:1319–1328
- . Altering pharmacokinetics of radiolabeled antibodies by the interposition of metabolizable linkages. Metabolizable linkers and pharmacokinetics of monoclonal antibodies. Q J Nucl Med. 2002;46:206–223
- . Reagents for astatination of biomolecules: 3. Comparison of closo-decaborate(2-) and closo-dodecaborate(2-) moieties as reactive groups for labeling with astatine-211. Bioconjug Chem. 2009;20:591–602
- . Chemistry of boranes: XXXI. 1,10-Bis(hydroxymethyl)octachlorodecaborate (2-). J Am Chem Soc. 1967;89:4850–4852
- . Physiology. In: Foster HL, Small JD, Fox JG editor. The Mouse in Biomedical Research. New York: Academic Press; 1983;p. 248–292
- . Chemistry of boranes: XXX. Carbonyl derivatives of B10H102− and B12H122−. J Am Chem Soc. 1967;89:4842–4850
- . Chemistry of boranes: XIX. Derivative chemistry of B10H10−2 and B12H12−2. J Am Chem Soc. 1964;86:3973–3983
- Biodistributions, myelosuppression and toxicities in mice treated with an anti-CD45 antibody labeled with the α-emitting radionuclides bismuth-213 or astatine-211. Cancer Res. 2009;69:2408–2415
- Reduction of background activities by introduction of a diester linkage between antibody and a chelate in radioimmunodetection of tumor. J Nucl Med. 1989;30:1693–1701
- . Enhanced kidney clearance with an ester-linked 99mTc-radiolabeled antibody Fab′-chelator conjugate. Bioconjug Chem. 1990;1:431–437
- A novel bifunctional metabolizable linker for the conjugation of antibodies with radionuclides. Bioconjug Chem. 1991;2:71–76
- Decreased kidney uptake of technetium-99m-labelled Fab′ fragments in ovarian carcinoma bearing nude mice using a cleavable chelator. Nucl Med Biol. 1994;21:17–24
- . Chelate radiochemistry: cleavable linkers lead to altered levels of radioactivity in the liver. Int J Cancer. 1988;2:99–102
- . Cathepsin substrates as cleavable peptide linkers in bioconjugates, selected from a fluorescence quench combinatorial library. Bioconjug Chem. 1998;9:618–626
- Development of tissue plasminogen activator specific “on demand cleavable” (odc) linkers for radioimmunotherapy by screening one-bead-one-compound combinatorial peptide libraries. Bioconjug Chem. 2007;18:175–182
- . Reversible covalent chemistry in drug delivery. Curr Drug Discov Technol. 2005;2:123–160
- . Polymeric anticancer drugs with pH-controlled activation. Adv Drug Deliv Rev. 2004;56:1023–1050
- . Drug-polymer conjugates containing acid cleavable bonds. Crit Rev Ther Drug Carrier Syst. 1999;16:245–288
- Aryldithioethyloxycarbonyl (Ardec): a new family of amine protecting groups removable under mild reducing conditions and their applications to peptide synthesis. Chemistry. 2006;12:3655–3671
- . Preparation of 131I-labelled m-iodohippuric acid and its behaviour in kidney function studies compared to o-iodohippuric acid. Int J Appl Radiat Isot. 1973;24:463–469
- . Lysosomotropic agents. Biochem Pharm. 1974;23:2495–2531
- . Antibody conjugates with morpholinodoxorubicin and acid-cleavable linkers. Bioconjug Chem. 1990;1:325–330
- New hydrazone derivatives of adriamycin and their immunoconjugates — a correlation between acid stability and cytotoxicity. Bioconjug Chem. 1991;2:133–141
PII: S0969-8051(09)00252-2
doi: 10.1016/j.nucmedbio.2009.10.004
© 2010 Elsevier Inc. All rights reserved.
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Nuclear Medicine and Biology
Volume 37, Issue 2
, Pages 167-178
, February 2010
