Nuclear Medicine and Biology
Volume 36, Issue 7 , Pages 749-757 , October 2009

In-depth evaluation of the cycloaddition–retro-Diels–Alder reaction for in vivo targeting with [111In]-DTPA-RGD conjugates

  • Peter Laverman

      Affiliations

    • Department of Nuclear Medicine, Radboud University Nijmegen Medical Centre, 6500 HB Nijmegen, The Netherlands
    • Corresponding Author InformationCorresponding author. Department of Nuclear Medicine, Radboud University Nijmegen Medical Centre, PO Box 9101, 6500 HB Nijmegen, The Netherlands. Tel.: +31 24 3615054; fax: +31 24 3618942.
  • ,
  • Silvie A. Meeuwissen

      Affiliations

    • Department of Nuclear Medicine, Radboud University Nijmegen Medical Centre, 6500 HB Nijmegen, The Netherlands
    • Institute for Molecules and Materials, Radboud University Nijmegen, 6500 GL Nijmegen, The Netherlands
  • ,
  • Sander S. van Berkel

      Affiliations

    • Institute for Molecules and Materials, Radboud University Nijmegen, 6500 GL Nijmegen, The Netherlands
  • ,
  • Wim J.G. Oyen

      Affiliations

    • Department of Nuclear Medicine, Radboud University Nijmegen Medical Centre, 6500 HB Nijmegen, The Netherlands
  • ,
  • Floris L. van Delft

      Affiliations

    • Institute for Molecules and Materials, Radboud University Nijmegen, 6500 GL Nijmegen, The Netherlands
  • ,
  • Floris P.J.T. Rutjes

      Affiliations

    • Institute for Molecules and Materials, Radboud University Nijmegen, 6500 GL Nijmegen, The Netherlands
  • ,
  • Otto C. Boerman

      Affiliations

    • Department of Nuclear Medicine, Radboud University Nijmegen Medical Centre, 6500 HB Nijmegen, The Netherlands

Received 22 October 2008 ,Revised 1 May 2009 ,Accepted 2 May 2009.

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PII: S0969-8051(09)00126-7

doi: 10.1016/j.nucmedbio.2009.05.001

Nuclear Medicine and Biology
Volume 36, Issue 7 , Pages 749-757 , October 2009