« Previous
Next »
Nuclear Medicine and Biology
Volume 36, Issue 5
, Pages 495-504
, July 2009
Cu(II) bis(thiosemicarbazone) radiopharmaceutical binding to serum albumin: further definition of species dependence and associated substituent effects
References
- . Species-dependent binding of copper(II) bis(thiosemicarbazone) radiopharmaceuticals to serum albumin. J Nucl Med. 1995;36:1451–1455
- . Species dependence of [64Cu]Cu-bis(thiosemicarbazone) radiopharmaceutical binding to serum albumins. Nucl Med Biol. 2008;35:281–286
- Basken N.E., Mathias C.J., Green M.A., Elucidation of the human serum albumin (HSA) binding site for the Cu-PTSM and Cu-ATSM radiopharmaceuticals. J Pharm Sci, [in press] (DOI:doi:10.1002/jps.21570).
- . Synthesis and evaluation of copper radiopharmaceuticals with mixed bis(thiosemicarbazone) ligands. Nucl Med Biol. 1999;26:551–554
- . Mixed bis(thiosemicarbazone) ligands for the preparation of copper radiopharmaceuticals; synthesis and evaluation of tetradentate ligands containing two dissimilar thiosemicarbazone functions. J Med Chem. 1997;40:132–136
- . The characterization of two specific drug binding sites on human serum albumin. Mol Pharmacol. 1975;11:824–832
- . Further characterization of two specific drug binding sites on human serum albumin. Mol Pharmacol. 1976;12:1052–1061
- . Practical aspects of the ligand-binding and enzymatic properties of human serum albumin. Biol Pharm Bull. 2002;25(6):695–704
- . The binding of drugs to blood plasma macromolecules: recent advances and therapeutic significance. In: Testa B editors. Advances in drug research. vol. 13:London: Academic Press; 1984;p. 59–94
- . Binding of drugs to serum albumin XI: the specificity of three binding sites as studied with albumin immobilized in microparticles. Mol Pharmacol. 1979;16:767–777
- In: Lenter C editors. Geigy scientific tables, Physical chemistry composition of blood hematology somatometric data. vol. 3:Basle, Switzerland: CIBA GEIGY; 1984;p. 136–139
- . All about albumin. San Diego (Calif): Academic Press; 1994;
- . A comparison of drug binding sites on mammalian serum albumins. Biochem Pharmacol. 1992;44(5):873–879
- . Comparison of the binding characteristics of serum albumins from various animal species. Dev Pharmacol Ther. 1990;15:106–111
- . Species differences of serum albumins I: drug binding sites. Pharm Res. 1997;14(11):1607–1612
- . Structure–activity relationships for metal-labeled blood flow tracers: comparison of keto aldehyde bis(thiosemicarbazone)copper(II) derivatives. J Med Chem. 1990;33:1764–1770
- http://www.elephants.com
- . In: Statistical inference. Pacific Grove (Calif): Duxbury; 2002;p. 240–245
- . The universal protein resource. Nucleic Acids Res. 2007;35:D193–D197http://www.uniprot.org
- . CLUSTAL W: improving the sensitivity of progressive multiple sequence alignment through sequence weighting, position-specific gap penalties and weight matrix choice. Nucleic Acids Res. 1994;22:4673–4680
- CLUSTAL W and CLUSTAL X version 2.0. Bioinformatics. 2007;23:2947–2948
- . Crystal structure of human serum albumin complexed with fatty acid reveals an asymmetric distribution of binding sites. Nat Struct Mol Biol. 1998;5:827–835
- . Crystal structure analysis of warfarin binding to human serum albumin. J Biol Chem. 2001;276:22804–22809
- . Structural basis of the drug-binding specificity of human serum albumin. J Mol Biol. 2005;353:38–52
- SAS, version 9.1.3. Cary (NC): SAS Institute Inc.; 2002–2003;
- . A new substituent constant, Π, derived from partition coefficients. J Am Chem Soc. 1964;86:5175–5180
PII: S0969-8051(09)00049-3
doi: 10.1016/j.nucmedbio.2009.02.006
© 2009 Elsevier Inc. All rights reserved.
« Previous
Next »
Nuclear Medicine and Biology
Volume 36, Issue 5
, Pages 495-504
, July 2009
