« Previous
Next »
Nuclear Medicine and Biology
Volume 34, Issue 8
, Pages 945-953
, November 2007
Gallium-68-labeled DOTA-rhenium-cyclized α-melanocyte-stimulating hormone analog for imaging of malignant melanoma
References
- . Analysis of the melanoma epidemic, both apparent and real: data from the 1973 through 1994 surveillance, epidemiology, and end results program registry. Arch Dermatol. 1999;135:275–280
- . Malignant melanoma of the skin. Epidemiology, risk factors, clinical diagnosis. Csa Lek Cesk. 1996;135:405–408
- . Radiolabeled alpha-melanocyte-stimulating hormone analogs for receptor-mediated targeting of melanoma: from tritium to indium. J Mol Recognit. 2003;16:248–254
- A fluorinated glucose analog, 2-fluoro-2-deoxy-d-glucose (F-18): nontoxic tracer for rapid tumor detection. J Nucl Med. 1980;21:670–675
- . Systematic review of the diagnostic accuracy of 18F-fluorodeoxyglucose positron emission tomography in melanoma patients. Cancer. 2001;91:1530–1542
- . Quantitative PET studies in pretreated melanoma patients: a comparison of 6-[18F]fluoro-l-DOPA with 18F-FDG and 15O-water using compartment and noncompartment analysis. J Nucl Med. 2001;42:248–256
- . Technetium-labeled monoclonal antibodies for imaging metastatic melanoma: results of a multicenter clinical study. Semin Oncol. 1988;15:608–618
- Radioimmunodetection of human melanoma with indium-111-labeled monoclonal antibody. J Nucl Med. 1988;29:329–337
- Characterization of a human–mouse chimeric antibody reactive with a human melanoma associated antigen. Prog Clin Biol Res. 1989;288:101–105
- . Amelanotic malignant melanoma. Semin Cutan Med Surg. 1997;16:122–130
- . The control of gene expression in melanocytes and melanomas. Melanoma Res. 1996;6:277–284
- . Melanoma: histological diagnosis and prognosis. New York: Raven; 1983;
- Biodistribution and pharmacokinetics of the alphavbeta3-selective tracer 18F-galacto-RGD in cancer patients. J Nucl Med. 2005;46:1333–1341
- . 3′-18F-Fluoro-3′-deoxy-l-thymidine: a new tracer for staging metastatic melanoma?. J Nucl Med. 2003;44:1927–1932
- Low efficacy of 18F-FDG PET for detection of uveal malignant melanoma compared with 123I-IMP SPECT. J Nucl Med. 2006;47:404–409
- 123I-N-(2-diethylaminoethyl)-2-iodobenzamide: a potential imaging agent for cutaneous melanoma staging. Eur J Nucl Med Mol Imaging. 2002;29:1478–1484
- Radioiodinated N-[3-(4-morpholino)propyl]-N-methyl-2-hydroxy-5-iodo-3-methylbenzylamine (ERC9): a new potential melanoma imaging agent. Eur J Nucl Med. 2001;28:408–417
- The melanocortin receptors: agonists, antagonists, and the hormonal control of pigmentation. Recent Prog Horm Res. 1996;51:287–317[discussion 318]
- Cloning and functional characterization of a family of receptors for the melanotropic peptides. Ann N Y Acad Sci. 1993;680:342–363
- . alpha-Melanocyte stimulating hormone, inflammation and human melanoma. Peptides. 2006;27:444–452
- Molecular cloning of a novel melanocortin receptor. J Biol Chem. 1993;268:8246–8250
- Molecular cloning, expression, and gene localization of a fourth melanocortin receptor. J Biol Chem. 1993;268:15174–15179
- . Cloning and expression of a new member of the melanocyte-stimulating hormone receptor family. J Mol Endocrinol. 1994;12:203–213
- . Molecular cloning, functional expression and pharmacological characterization of a mouse melanocortin receptor gene. Biochem J. 1994;299:367–373
- . Molecular cloning of a mouse melanocortin 5 receptor gene widely expressed in peripheral tissues. Biochemistry. 1994;33:4543–4549
- . In: Cone RD editors. Propiomelanocortin and the melanocortin peptides. Totowa, New Jersey: Humana Press; 2000;p. 3–67
- Interaction of an alpha-melanocyte-stimulating hormone-diphtheria toxin fusion protein with melanotropin receptors in human melanoma metastases. Cancer Res. 1992;52:2545–2548
- Melanotropin receptors demonstrated in situ in human melanoma. J Clin Invest. 1990;85:1825–1832
- Characterization of receptors for alpha-melanocyte-stimulating hormone on human melanoma cells. Cancer Res. 1989;49:6352–6358
- . Evaluation of the human melanoma targeting properties of radiolabeled α-melanocyte stimulating hormone peptide analogues. Bioconjug Chem. 2003;14:1177–1184
- . In vivo evaluation of 99mTc/188Re-labeled linear alpha-melanocyte stimulating hormone analogs for specific melanoma targeting. Nucl Med Biol. 1999;26:687–693
- . 64Cu-labeled alpha-melanocyte-stimulating hormone analog for microPET imaging of melanocortin 1 receptor expression. Bioconjug Chem. 2007;18:765–772
- Small-animal PET of melanocortin 1 receptor expression using a 18F-labeled a-melanocyte-stimulating hormone analog. J Nucl Med. 2007;48:987–994
- A gallium-labeled DOTA-alpha-melanocyte-stimulating hormone analog for PET imaging of melanoma metastases. J Nucl Med. 2004;45:116–123
- . DOTA a-melanocyte-stimulating hormone analogues for imaging metastatic melanoma lesions. Ann N Y Acad Sci. 2003;994:378–383
- . Melanoma targeting with DOTA-melanocyte-stimulating hormone analogs: structural parameters affecting tumor uptake and kidney uptake. J Nucl Med. 2005;46:887–895
- . A novel DOTA-alpha-melanocyte-stimulating hormone analog for metastatic melanoma diagnosis. J Nucl Med. 2002;43:1699–1706
- Evaluation of an 111In-DOTA-rhenium cyclized alpha-MSH analog: a novel cyclic-peptide analog with improved tumor-targeting properties. J Nucl Med. 2001;42:1847–1855
- . Radioiodination of rhenium cyclized alpha-melanocyte-stimulating hormone resulting in enhanced radioactivity localization and retention in melanoma. Cancer Res. 2004;64:1411–1418
- . Imaging of melanoma using 64Cu- and 86Y-DOTA-ReCCMSH(Arg11), a cyclized peptide analogue of alpha-MSH. J Med Chem. 2005;48:2985–2992
- . Copper radionuclides and radiopharmaceuticals in nuclear medicine. Nucl Med Biol. 1996;23:957–980
- Efficient production of high specific activity 64Cu using a biomedical cyclotron. Nucl Med Biol. 1997;24:35–43
- Preparation of high specific activity 86Y using a small biomedical cyclotron. Nucl Med Biol. 2005;32:891–897
- . 68Ga-labeled peptides in tumor imaging. J Nucl Med. 2005;46:172S–178S
- Performance evaluation of the microPET Focus: a third-generation microPET scanner dedicated to animal imaging. J Nucl Med. 2005;46:455–463
- Synthesis and biological evaluation of Cu-64 labeled rhenium-cyclized a-MSH peptide analog using a cross-bridged cyclam chelator. J Nucl Med. 2007;48:64–72
- Structure–activity relationships of [Nle4, d-Phe7]alpha-MSH. Discovery of a tripeptidyl agonist exhibiting sustained bioactivity. Ann N Y Acad Sci. 1993;680:597–599
- 4-Norleucine, 7-d-phenylalanine-alpha-melanocyte-stimulating hormone: a highly potent alpha-melanotropin with ultralong biological activity. Proc Natl Acad Sci U S A. 1980;77:5754–5758
- . Cyclic melanotropins. 9. 7-d-Phenylalanine analogues of the active-site sequence. J Med Chem. 1985;28:583–588
- . Potent and prolonged acting cyclic lactam analogues of alpha-melanotropin: design based on molecular dynamics. J Med Chem. 1989;32:2555–2561
- Cyclic lactam alpha-melanotropin analogues of Ac-Nle4-cyclo[Asp5, d-Phe7,Lys10] alpha-melanocyte-stimulating hormone-(4–10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors. J Med Chem. 1995;38:3454–3461
- . Design and characterization of alpha-melanotropin peptide analogs cyclized through rhenium and technetium metal coordination. Proc Natl Acad Sci U S A. 1998;95:12814–12818
- . Melanoma-targeting properties of (99m)technetium-labeled cyclic alpha-melanocyte-stimulating hormone peptide analogues. Cancer Res. 2000;60:5649–5658
- . In vivo evaluation of 188Re-labeled alpha-melanocyte stimulating hormone peptide analogs for melanoma therapy. Int J Cancer. 2002;101:480–487
- . Tumor targeting properties of 90Y and 177Lu labeled alpha-melanocyte stimulating hormone peptide analogues in a murine melanoma model. Nucl Med Biol. 2005;32:485–493
- Cu-64-TETA-octreotide as a PET imaging agent for patients with neuroendocrine tumors. J Nucl Med. 2001;42:213–221
- PET imaging of somatostatin receptors using [68GA]DOTA-d-Phe1-Tyr3-octreotide: first results in patients with meningiomas. J Nucl Med. 2001;42:1053–1056
- 86Y-DOTA-d-Phe1-Tyr3-octreotide (SMT487)—a phase 1 clinical study: pharmacokinetics, biodistribution and renal protective effect of different regimens of amino acid co-infusion. Eur J Nucl Med Mol Imaging. 2003;30:510–518
- Preparation and biological evaluation of copper-64-labeled Tyr3-octreotate using a cross-bridged macrocyclic chelator. Clin Cancer Res. 2004;10:8674–8682
- Comparative in vivo stability of copper-64-labeled cross-bridged and conventional tetraazamacrocyclic complexes. J Med Chem. 2004;47:1465–1474
- Comparison of four bifunctional chelates for radiolabeling monoclonal antibodies with copper radioisotopes: biodistribution and metabolism. Bioconjug Chem. 1996;7:511–522
- The in vivo behavior of copper-64-labeled azamacrocyclic complexes. Nucl Med Biol. 1998;25:523–530
- Radiometal-labelled macrocyclic chelator-derivatised somatostatin analogue with superb tumour-targeting properties and potential for receptor-mediated internal radiotherapy. Chem Eur J. 1999;5:1974–1981
- . Radiolabelling DOTA-peptides with 68Ga. Eur J Nucl Med Mol Imaging. 2005;32:478–485
- . 68Ga-labelled DOTA-derivatised peptide ligands. Eur J Nucl Med Mol Imaging. 2004;31:1097–1104
- d-Lysine reduction of indium-111 octreotide and yttrium-90 octreotide renal uptake. J Nucl Med. 1997;38:1929–1933
PII: S0969-8051(07)00183-7
doi: 10.1016/j.nucmedbio.2007.07.003
© 2007 Elsevier Inc. All rights reserved.
« Previous
Next »
Nuclear Medicine and Biology
Volume 34, Issue 8
, Pages 945-953
, November 2007
