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Nuclear Medicine and Biology
Volume 34, Issue 7
, Pages 823-831
, October 2007
Imaging multidrug resistance with 4-[18F]fluoropaclitaxel
References
- . Multidrug resistance transporters and modulation. Curr Opin Oncol. 2000;12:450–458
- . How cancer-cells evade chemotherapy — 16th Richard-and-Hinda-Rosenthal-Foundation Award Lecture. Cancer Res. 1993;53:747–754
- . MDR expression in normal-tissues — pharmacological implications for the clinical use of P-glycoprotein inhibitors. Hematol Oncol Clin North Am. 1995;9:319–336
- . Detection of P-glycoprotein with 4 monoclonal-antibodies in normal and tumor-tissues. Arch Otolaryngol Head Neck Surg. 1993;119:753–757
- Role of intestinal P-glycoprotein (mdr1) in interpatient variation in the oral bioavailability of cyclosporine. Clin Pharmacol Ther. 1997;62:248–260
- . The barrier function of CYP3A4 and P-glycoprotein in the small bowel. Adv Drug Deliv Rev. 1997;27:161–170
- . Multidrug transporters as drug targets. Curr Drug Targets. 2006;7:911–921
- . Kinetic parameters for reversal of the multidrug pump as measured for drug accumulation and cell killing. Cancer Chemother Pharmacol. 1996;38:181–190
- . Effects of MDR reversing agent combinations on the H-3-daunomycin accumulation in drug-sensitive and drug-resistant human cancer cells. Anticancer Res. 2000;20:2617–2623
- Identification of a multidrug-resistance modulator with clinical potential by analysis of synergistic activity in-vitro, toxicity in-vivo and growth delay in a solid human tumor xenograft. Biochem Pharmacol. 1994;47:257–266
- . Visualization of multidrug resistance in vivo. Eur J Nucl Med. 1999;26:283–293
- . Differential-effects of P-glycoprotein inhibitors on Nih3t3 cells transfected with wild-type (G185) or mutant (V185) multidrug transporters. Cancer Res. 1995;55:1086–1091
- Fractional retention of technetium-99m-sestamibi as an index of P-glycoprotein expression in untreated breast cancer patients. J Nucl Med. 1997;38:1348–1351
- . Modulation and prevention of multidrug resistance by inhibitors of P-glycoprotein. Cancer Chemother Pharmacol. 1997;40:S13–S19
- Fractional retention of 99mTc-MIBI and proliferation in untreated breast cancer. Eur J Nucl Med. 1999;26:PS455
- . Scintigraphic prediction of resistance to radiation and chemotherapy in patients with lung carcinoma — technetium 99m-tetrofosmin and thallium-201 dual single photon emission computed tomography study. Cancer. 1999;86:1470–1479
- . Characterization of P-glycoprotein transport and inhibition in vivo. Cancer Res. 1998;58:276–282
- Detection of in vivo P-glycoprotein inhibition by PSC 833 using Tc-99m sestamibi. Clin. Cancer Res. 1997;3:545–552
- . In vivo measurement of [C-11] verapamil kinetics in human tissues. Eur J Clin Pharmacol. 2001;56:827–829
- Evaluation of C-11-colchicine for PET imaging of multiple drug resistance. J Nucl Med. 2000;41:493–501
- Carbon-11-labeled daunorubicin and verapamil for probing P-glycoprotein in tumors with PET. J Nucl Med. 1996;37:1571–1575
- Complete in vivo reversal of P-glycoprotein pump function in the blood–brain barrier visualized with positron emission tomography. Br J Pharmacol. 1998;124:1413–1418
- A new in vivo method to study P-glycoprotein transport in tumors and the blood–brain barrier. Cancer Res. 1999;59:2411–2416
- Radiosynthesis of [C-11] paclitaxel. J Labelled Compd Radiopharm. 2002;45:471–477
- Radiosynthesis of [C-11] docetaxel. J Labelled Compd Radiopharm. 2004;47:763–777
- . 18F-labeled fluorouracil positron emission tomography and the prognoses of colorectal carcinoma patients with metastases to the liver treated with 5-fluorouracil. Cancer. 1998;83:245–253
- . Perfusion of colorectal liver metastases and uptake of fluorouracil assessed by H2(15)O and [18F]uracil positron emission tomography (PET). Eur J Cancer. 1993;29A:1682–1686
- . Preclinical pharmacokinetics of paclitaxel and docetaxel. Anticancer Drugs. 1998;9:1–17
- Co-expression of several molecular mechanisms of multidrug resistance and their significance for paclitaxel cytotoxicity in human AML HL-60 cells. Leukemia. 1997;11:253–257
- Monitoring tumor glucose utilization by positron emission tomography for the prediction of treatment response to epidermal growth factor receptor kinase inhibitors. Clin Cancer Res. 2006;12:5659–5667
- P-glycoprotein expression is associated with FDG uptake and cell differentiation in patients with untreated lung cancer. Nucl Med Commun. 2004;25:19–27
- Synthesis, biodistribution and imaging properties of indium-111–DTPA–paclitaxel in mice bearing mammary tumors. J Nucl Med. 1997;38:1042–1047
- Estimation of paclitaxel biodistribution and uptakein human-derived xenografts in vivo with (18)F-fluoropaclitaxel. J Nucl Med. 2005;46:1866–1871
- Predicting chemotherapy response to paclitaxel with 18F-fluoropaclitaxel and PET. J Nucl Med. 2006;47:1995–1999
- . Pharmacological insights from P-glycoprotein knockout mice. Int J Clin Pharmacol Ther. 1998;36:9–13
- . Comparison of the biodistribution of fluorinated and tritiated paclitaxel (PAC) in mdr1a(−)/1b(−) knockout vs. wildtype mice. J Nucl Med. 2002;43:277P
- . Radiochemical synthesis of [18F]fluoropaclitaxel ([18F]FPAC). J Labelled Compd Radiopharm. 2001;S903–S905
- . Biodistribution, radiation dose estimates and Pgp modulation studies of [18F]paclitaxel. J Nucl Med. 2001;42(S):279P
- . Automated synthesis of 18F analogue of paclitaxel (PAC): [18F]paclitaxel (FPAC). Appl Radiat Isot. 2007;65:696–700
- . Genetic risk profiles for cancer susceptibility and therapy response. Recent Results Cancer Res. 2007;174:19–36
- Inclusion of taxanes, particularly weekly paclitaxel, in preoperative chemotherapy improves pathologic complete response rate in estrogen receptor-positive breast cancers. Ann Oncol. 2007;18:874–880
- Prognostic relevance of response evaluation using [F-18]-2-fluoro-2-deoxy-d-glucose positron emission tomography in patients with locally advanced non-small-cell lung cancer. J Clin Oncol. 2005;23:8362–8370
- Early response monitoring by FOG-PET to neoadjuvant chemotherapy in locally advanced breast cancer patients. J Clin Oncol. 2005;23:140S
- . Early prediction of response to chemotherapy in metastatic breast cancer using sequential F-18-FDG PET. J Nucl Med. 2005;46:1144–1150
PII: S0969-8051(07)00124-2
doi: 10.1016/j.nucmedbio.2007.04.011
© 2007 Elsevier Inc. All rights reserved.
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Nuclear Medicine and Biology
Volume 34, Issue 7
, Pages 823-831
, October 2007
