« Previous
Next »
Nuclear Medicine and Biology
Volume 33, Issue 4
, Pages 513-520
, May 2006
Rhemium-186-monoaminemonoamidedithiol-conjugated bisphosphonate derivatives for bone pain palliation
References
- . Osteolytic bone metastasis in breast cancer. Breast Cancer Res Treat. 1994;32:73–84
- . Malignant bone pain: pathophysiology and treatment. Pain. 1997;69:1–18
- . Single-dose radiotherapy (6 Gy): palliation in painful bone metastases. Radiother Oncol. 1995;36:198–202
- . Radiopharmaceutical therapy for palliation of bone pain from osseous metastases. J Nucl Med. 2004;45:1358–1365
- . Use of radionuclides for the palliation of bone metastases. Semin Radiat Oncol. 2000;10:103–114
- . Studies of the structure and composition of rhenium-1,1-hydroxyethylidenediphosphonate (HEDP) analogues of the radiotherapeutic agent (186)ReHEDP. Inorg Chem. 1997;36:3055–3063
- . Evaluation of toxicity and efficacy of 186Re-hydroxyethylidene diphosphonate in patients with painful bone metastases of prostate or breast cancer. J Nucl Med. 2000;41:1689–1694
- Palliative therapy using rhenium-186-HEDP in painful breast osseous metastases. Anticancer Res. 1997;17:1767–1772
- High activity rhenium-186 HEDP with autologous peripheral blood stem cell rescue: a phase I study in progressive hormone refractory prostate cancer metastatic to bone. Br J Cancer. 2002;86:1715–1720
- . Visualization of the stomach on rhenium-186 HEDP imaging after therapy for metastasized prostate carcinoma. Clin Nucl Med. 1999;24:898–899
- . Pharmacokinetics of rhenium-186 after administration of rhenium-186-HEDP to patients with bone metastases. J Nucl Med. 1992;33:646–651
- Synthesis and biodistribution studies of 186Re complex of 1-hydroxyethylidene-1,1-diphosphonate for treatment of painful osseous metastases. Radioisotopes. 1995;44:514–522
- Design of a radiopharmaceutical for the palliation of painful bone metastases: rhenium-186-labeled bisphosphonate derivative. J Label Cmpd Radiopharm. 2004;47:753–761
- . The influence of multidentate organic phosphonates on the crystal growth of hydroxyapatite. Calcif Tissue Res. 1973;13:295–303
- . Structural requirements for bisphosphonate actions in vitro. J Bone Miner Res. 1994;9:1875–1882
- . Production of 186/188Re and recovery of tungsten from spent 188W/188Re generator. Radiochemistry. 2000;42:551–554
- Kieczykowski GR. New process for preparing an antihypercalcemic agent. UK Patent GB 2248061A, 1992.
- . Selective drug delivery system to bone: small peptide (Asp)6 conjugation. J Bone Miner Res. 2000;15:936–943
- . Preferential adsorption of dentin and bone acidic proteins on the (100) face of hydroxyapatite crystals. Biochim Biophys Acta. 1991;1075:56–60
- Radiation dose estimates of 186Re-hydroxyethylidene diphosphonate for palliation of metastatic osseous lesions: an animal model study. Nucl Med Commun. 1997;18:582–588
- . Bisphosphonates: mechanisms of action. Endocr Rev. 1998;19:80–100
- . Bisphosphonates: mechanisms of action. J Clin Invest. 1996;97:2692–2696
- . Calcium affinity of coordinated diphosphonate ligands. Single-crystal structure of [(en)2Co(O2P(OH)CH2P(OH)O2]ClO4·H2O. Implications for the chemistry of technetium-99m-diphosphonate skeletal imaging agents. Inorg Chem. 1983;22:1332–1338
- . New diphosphonate compounds for skeletal imaging: comparison with methylene diphosphonate. Radiology. 1983;149:823–828
- . A comparison of skeletal uptakes of three diphosphonates by whole-body retention: concise communication. J Nucl Med. 1981;22:880–883
- . Skeletal localization of samarium-153 chelates: potential therapeutic bone agents. J Nucl Med. 1987;28:495–504
- . 153Sm-EDTMP and 186Re-HEDP as bone therapeutic radiopharmaceuticals. Int J Rad Appl Instrum B. 1987;14:223–232
PII: S0969-8051(06)00062-X
doi: 10.1016/j.nucmedbio.2006.03.006
© 2006 Elsevier Inc. All rights reserved.
« Previous
Next »
Nuclear Medicine and Biology
Volume 33, Issue 4
, Pages 513-520
, May 2006
